Please use this identifier to cite or link to this item:
https://hdl.handle.net/2440/123184
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Full metadata record
DC Field | Value | Language |
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dc.contributor.author | Reekie, T.A. | - |
dc.contributor.author | Wilkinson, S.M. | - |
dc.contributor.author | Law, V. | - |
dc.contributor.author | Hibbs, D.E. | - |
dc.contributor.author | Ong, J.A. | - |
dc.contributor.author | Kassiou, M. | - |
dc.date.issued | 2017 | - |
dc.identifier.citation | Organic and Biomolecular Chemistry, 2017; 15(3):576-580 | - |
dc.identifier.issn | 1477-0520 | - |
dc.identifier.issn | 1477-0539 | - |
dc.identifier.uri | http://hdl.handle.net/2440/123184 | - |
dc.description | Published on 14 December 2016. | - |
dc.description.abstract | Preparation of N-(indol-2-yl)amides and N-(indol-3-yl)amides are scarce in the scientific literature due to unstable intermediates impeding current reported syntheses. We have employed cheap and readily available substrates in the Curtius rearrangement of indole-3-carboxazide to afford N-(indol-3-yl)amides. The reaction is observed for alkyl and aryl carboxylic acids and both N-substituted or 1H-indole derivatives are tolerated. This approach was extended to the preparation of N-(indol-2-yl)amides from the corresponding indole-2-carboxazides. | - |
dc.description.statementofresponsibility | Tristan A. Reekie, Shane M. Wilkinson, Vivian Law, David E. Hibbs, Jennifer A. Ong and Michael Kassiou | - |
dc.language.iso | en | - |
dc.publisher | Royal Society of Chemistry | - |
dc.rights | This journal is © The Royal Society of Chemistry 2017. Open Access Article. This article is licensed under a Creative Commons Attribution-NonCommercial 3.0 Unported Licence. | - |
dc.source.uri | http://dx.doi.org/10.1039/c6ob02622b | - |
dc.title | Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores | - |
dc.type | Journal article | - |
dc.identifier.doi | 10.1039/c6ob02622b | - |
dc.relation.grant | http://purl.org/au-research/grants/nhmrc/1037979 | - |
pubs.publication-status | Published | - |
dc.identifier.orcid | Ong, J.A. [0000-0002-0958-460X] | - |
Appears in Collections: | Aurora harvest 4 Physiology publications |
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hdl_123184.pdf | Published version | 394.53 kB | Adobe PDF | View/Open |
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