Formulation effects in percutaneous absorption

dc.contributor.authorKuswahyuning, R.
dc.contributor.authorGrice, J.E.
dc.contributor.authorMoghimi, H.R.
dc.contributor.authorRoberts, M.S.
dc.contributor.editorDragicevic, N.
dc.contributor.editorMaibach, H.I.
dc.date.issued2015
dc.description.abstractFormulation optimisation is one of the strategies used for optimising delivery into or through the skin. In addition to ensuring that an active chemical is delivered at an adequate rate to achieve therapeutic concentrations over the intended duration, physicochemical formulation stability as well as product acceptance must also be achieved. There is a continual growth in new potential delivery systems, such as microemulsions, liposomes, ultradeformable liposomes and lipid nanoparticles, offering various advantages, either for dermal and transdermal delivery. However, choosing and designing the most suitable formulation system for a given compound is a complex process. In this chapter, various aspects of formulation-related transdermal drug delivery are discussed and an alternative approach to the design of formulation systems is reviewed. In addition, current formulation-based strategies and the effects of commonly added ingredients for stability and aesthetic purposes are covered. Finally, formulations based on some novel delivery systems are discussed.
dc.identifier.citationSource details - Title: Percutaneous penetration enhancers chemical methods in penetration enhancement : drug manipulation strategies and vehicle effects, 2015 / Dragicevic, N., Maibach, H.I. (ed./s), Ch.9, pp.109-134
dc.identifier.doi10.1007/978-3-662-45013-0_9
dc.identifier.isbn9783662450123
dc.identifier.urihttps://hdl.handle.net/11541.2/116334
dc.language.isoen
dc.publisherSpringer
dc.publisher.placeBerlin
dc.relation.fundingNHMRC 1002611
dc.rightsCopyright 2015 Springer-Verlag Berlin Heidelberg
dc.source.urihttps://doi.org/10.1007/978-3-662-45013-0_9
dc.subjectskin
dc.subjecttransdermal drug delivery
dc.subjectformulation optimisation
dc.subjectformulation effects
dc.subjectpercutaneous absorption
dc.titleFormulation effects in percutaneous absorption
dc.typeBook chapter
pubs.publication-statusPublished
ror.mmsid9915989011201831

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